-Dale L Boger Researcher Activity Profile

Research Author Detailed Information 

Dale L Boger Publication Rate By Year

Dale L Boger has published 1 paper(s) in 2002, 2 paper(s) in 2003, 5 paper(s) in 2004, 1 paper(s) in 2005, 6 paper(s) in 2006, 10 paper(s) in 2007, 5 paper(s) in 2008, for a total of 30 research publications in total.

Dale L Dl Boger Author Information

LAST NAME: boger

FIRST NAME: Dale L

INITIALS: dl

AFFILIATION:

Papers

Dale L Boger's Publication Record

1. Structure-based design, synthesis, evaluation, and crystal structures of transition state analogue inhibitors of inosine monophosphate cyclohydrolase. Year Published: 2007
Department of Molecular Biology, The Scripps Research Institute, La Jolla, California 92037, USA.
2. Intramolecular diels-alder/1,3-dipolar cycloaddition cascade of 1,3,4-oxadiazoles. Year Published: 2006
Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
3. Total synthesis of (-)- and ent-(+)-vindoline and related alkaloids. Year Published: 2006
Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
4. Total synthesis of piericidin A1 and B1 and key analogues. Year Published: 2006
Departments of Chemistry and Molecular and Experimental Medicine, and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, La Jolla, California 92037, USA.
5. Delineation of a fundamental alpha-ketoheterocycle substituent effect for use in the design of enzyme inhibitors. Year Published: 2006
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, CA 92037, USA.
6. Asymmetric total synthesis of (+)- and ent-(-)-yatakemycin and duocarmycin SA: evaluation of yatakemycin key partial structures and its unnatural enantiomer. Year Published: 2006
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, La Jolla, California 92037, USA.
7. Potent and selective alpha-ketoheterocycle-based inhibitors of the anandamide and oleamide catabolizing enzyme, fatty acid amide hydrolase. Year Published: 2007
Department of Chemistry, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
8. Structure-activity relationships of alpha-ketooxazole inhibitors of fatty acid amide hydrolase. Year Published: 2007
Department of Chemistry, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
9. Alanine scan of [L-Dap(2)]ramoplanin A2 aglycon: assessment of the importance of each residue. Year Published: 2007
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
10. Total synthesis, stereochemical reassignment, and absolute configuration of chlorofusin. Year Published: 2007
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, CA 92037, USA.
11. Systematic exploration of the structural features of yatakemycin impacting DNA alkylation and biological activity. Year Published: 2007
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
12. Rational design, synthesis, and evaluation of key analogues of CC-1065 and the duocarmycins. Year Published: 2007
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
13. A unique class of duocarmycin and CC-1065 analogues subject to reductive activation. Year Published: 2007
Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
14. Direct coupling of catharanthine and vindoline to provide vinblastine: total synthesis of (+)- and ent-(-)-vinblastine. Year Published: 2008
Department of Chemistry and Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
15. Rational design, synthesis, and evaluation of key analogues of CC-1065 and the duocarmycins. Year Published: 2007
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
16. Intramolecular Diels-Alder and tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition reactions of 1,3,4-oxadiazoles. Year Published: 2002
Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
17. Partitioning the loss in vancomycin binding affinity for D-Ala-D-Lac into lost H-bond and repulsive lone pair contributions. Year Published: 2003
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
18. Fundamental role of the fostriecin unsaturated lactone and implications for selective protein phosphatase inhibition. Year Published: 2003
Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
19. Establishing the parabolic relationship between reactivity and activity for derivatives and analogues of the duocarmycin and CC-1065 alkylation subunits. Year Published: 2004
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
20. Total synthesis and examination of three key analogues of ramoplanin: a lipoglycodepsipeptide with potent antibiotic activity. Year Published: 2004
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
21. Dissecting ramoplanin: mechanistic analysis of synthetic ramoplanin analogues as a guide to the design of improved antibiotics. Year Published: 2004
Department of Chemistry, Princeton University, Princeton, New Jersey 08544, USA.
22. Total synthesis, structure revision, and absolute configuration of (+)-yatakemycin. Year Published: 2004
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
23. A powerful selection assay for mixture libraries of DNA alkylating agents. Year Published: 2004
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
24. Total synthesis of piericidin A1 and B1. Year Published: 2005
Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
25. Delineation of a fundamental alpha-ketoheterocycle substituent effect for use in the design of enzyme inhibitors. Year Published: 2006
Department of Chemistry and the Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, CA 92037, USA.
26. A unique class of duocarmycin and CC-1065 analogues subject to reductive activation. Year Published: 2007
Department of Chemistry and The Skaggs Institute for Chemical Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.
27. Optimization of alpha-Ketooxazole Inhibitors of Fatty Acid Amide Hydrolase. Year Published: 2008
boger@scripps.edu.
28. Disruption of the MYC transcriptional function by a small-molecule antagonist of MYC/MAX dimerization. Year Published: 2008
Northern Institute for Cancer Research, Newcastle University, Newcastle upon Tyne, NE2 4HH, UK.
29. Disruption of the MYC transcriptional function by a small-molecule antagonist of MYC/MAX dimerization. Year Published: 2008
Northern Institute for Cancer Research, Newcastle University, Newcastle upon Tyne, NE2 4HH, UK.
30. Optimization of alpha-ketooxazole inhibitors of fatty acid amide hydrolase. Year Published: 2008
Department of Chemistry, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037, USA.