-Jan Balzarini Researcher Activity Profile

Research Author Detailed Information 

Jan Balzarini Publication Rate By Year

Jan Balzarini has published 52 paper(s) in 2007, 6 paper(s) in 2008, for a total of 58 research publications in total.

Jan J Balzarini Author Information

LAST NAME: balzarini

FIRST NAME: jan

INITIALS: J

AFFILIATION:

Papers

Jan Balzarini's Publication Record

1. Syntheses and anti-HIV activities of (+/-)-norcarbovir and (+/-)-norabacavir. Year Published: 2007
Department of Chemistry & Biochemistry, University of Notre Dame, 251 Nieuwland Science Hall, Notre Dame, Indiana 46556, USA.
2. Antiviral activity of triazine analogues of 1-(S)-[3-hydroxy-2-(phosphonomethoxy)propyl]cytosine (cidofovir) and related compounds. Year Published: 2007
Gilead Sciences & IOCB Research Centre, Centre for New Antivirals and Antineoplastics (IOCB), Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic. marcela@uochb.cas.cz
3. Synthesis, structural characterization, and biological studies of new antimony(III) complexes with thiones. The influence of the solvent on the geometry of the complexes. Year Published: 2007
Section of Inorganic and Analytical Chemistry, Department of Chemistry, University of Ioannina, 45110 Ioannina, Greece.
4. Cytostatic activity of novel 4'-aminochalcone-based imides. Year Published: 2007
Department of Chemistry, Acadia University, Wolfville, NS, Canada B4P 2R6. ajha@acadiau.ca
5. Entry of hepatitis C virus and human immunodeficiency virus is selectively inhibited by carbohydrate-binding agents but not by polyanions. Year Published: 2007
Department of Microbiology and Immunology, Albert Einstein College of Medicine, Bronx, New York, USA.
6. Synthesis, anticancer, and cytotoxic activities of some mononuclear Ru(II) compounds. Year Published: 2007
Department of Pharmaceutical Chemistry, KLES College of Pharmacy, 2nd Block, Rajajinagar, Bangalore 560010, Karnataka, India. subhasskarki@hotmail.com
7. Design, synthesis, and cytostatic activity of novel cyclic curcumin analogues. Year Published: 2007
8. Efficient conversion of tetrapeptide-based TSAO prodrugs to the parent drug by dipeptidyl-peptidase IV (DPPIV/CD26). Year Published: 2007
9. Characterization and structural analysis of novel mutations in human immunodeficiency virus type 1 reverse transcriptase involved in the regulation of resistance to nonnucleoside inhibitors. Year Published: 2007
Department of Experimental Medicine, University of Rome Tor Vergata, Via Montpellier 1, 00133 Rome, Italy. ceccherini@med.uniroma2.it
10. Synthesis and biological evaluation of 2-amino-3-(3', 4', 5'-trimethoxy-phenylsulfonyl)-5-aryl thiophenes as a new class of antitubulin agents. Year Published: 2007
11. Synthesis, structural characterization, and biological studies of new antimony(III) complexes with thiones. The influence of the solvent on the geometry of the complexes. Year Published: 2007
Section of Inorganic and Analytical Chemistry, Department of Chemistry, University of Ioannina, 45110 Ioannina, Greece.
12. Rational design of 5'-thiourea-substituted alpha-thymidine analogues as thymidine monophosphate kinase inhibitors capable of inhibiting mycobacterial growth. Year Published: 2007
Laboratory for Medicinal Chemistry (FFW), University of Gent, Harelbekestraat 72, 9000 Ghent, Belgium.
13. Targeting platelet-derived endothelial cell growth factor/thymidine phosphorylase for cancer therapy. Year Published: 2007
Laboratory of Virology and Chemotherapy, Rega Institute for Medical Research, K.U. Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium. sandra.liekens@rega.kuleuven.be
14. Ester prodrugs of cyclic 1-(S)- [3-hydroxy-2-(phosphonomethoxy)propyl]-5-azacytosine: synthesis and antiviral activity. Year Published: 2007
Gilead Sciences and IOCB Research Centre, Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic. marcela@uochb.cas.cz
15. Hydantoin derivatives of L- and D-amino acids: synthesis and evaluation of their antiviral and antitumoral activity. Year Published: 2007
Department of Medicinal Chemistry, Faculty of Pharmacy and Biochemistry, A. Kovaci?a 1, HR-10000 Zagreb, Croatia. zrajic@pharma.hr
16. Preclinical development of bicyclic nucleoside analogues as potent and selective inhibitors of varicella zoster virus. Year Published: 2007
Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK.
17. Mitochondrial expression of the Drosophila melanogaster multisubstrate deoxyribonucleoside kinase. Year Published: 2007
Karolinska Institute, Department of Laboratory Medicine, Division of Clinical Virology F68, S-14186 Stockholm, Sweden. nicola.solaroli@ki.se
18. Synthesis and biological evaluation of 2-amino-3-(3', 4', 5'-trimethoxy-phenylsulfonyl)-5-aryl thiophenes as a new class of antitubulin agents. Year Published: 2007
19. Rational design of 5'-thiourea-substituted alpha-thymidine analogues as thymidine monophosphate kinase inhibitors capable of inhibiting mycobacterial growth. Year Published: 2007
Laboratory for Medicinal Chemistry (FFW), University of Gent, Harelbekestraat 72, 9000 Ghent, Belgium.
20. New Developments of the "Lock-in" Modified cycloSal-d4TMPs. Year Published: 2007
Department of Chemistry, Organic Chemistry, Faculty of Science, University of Hamburg, Hamburg, Germany.
21. Alkyne-azide click chemistry mediated carbanucleosides synthesis. Year Published: 2007
22. Cross-metathesis mediated synthesis of new acyclic nucleoside phosphonates. Year Published: 2007
23. Antiviral Activity of 3-(3,5-Dimethylbenzyl)Uracil Derivatives Against Hiv-1 and HCMV. Year Published: 2007
Faculty of Pharmaceutical Sciences at Kagawa Campus, Tokushima Bunri University, Kagawa, Japan.
24. Novel non-nucleoside human cytomegalovirus inhibitors based upon tsao nucleoside derivatives: structure-activity relationships. Year Published: 2007
25. Design, synthesis, and cytostatic activity of novel cyclic curcumin analogues. Year Published: 2007
26. Efficient synthesis and in vitro cytostatic activity of 4-substituted triazolyl-nucleosides. Year Published: 2007
27. A p-[(18)F]Fluoroethoxyphenyl Bicyclic Nucleoside Analogue as a Potential Positron Emission Tomography Imaging Agent for Varicella-Zoster Virus Thymidine Kinase Gene Expression. Year Published: 2007
guy.bormans@pharm.kuleuven.be.
28. Synthesis and Antiviral Activity of the Carbocyclic Analogue of the Highly Potent and Selective Anti-VZV Bicyclo Furano Pyrimidines. Year Published: 2007
mcguigan@cardiff.ac.uk.
29. Synthesis, structural characterization, and biological studies of new antimony(III) complexes with thiones. The influence of the solvent on the geometry of the complexes. Year Published: 2007
Section of Inorganic and Analytical Chemistry, Department of Chemistry, University of Ioannina, 45110 Ioannina, Greece.
30. New developments of the "lock-in" modified cycloSal-d4TMPs. Year Published: 2007
Department of Chemistry, Organic Chemistry, Faculty of Science, University of Hamburg, Martin Luther King-Platz 6, 20146 Hamburg, Germany.
31. Alkyne-azide click chemistry mediated carbanucleosides synthesis. Year Published: 2007
32. Cross-metathesis mediated synthesis of new acyclic nucleoside phosphonates. Year Published: 2007
33. Antiviral activity of 3-(3,5-dimethylbenzyl)uracil derivatives against HIV-1 and HCMV. Year Published: 2007
Faculty of Pharmaceutical Sciences at Kagawa Campus, Tokushima Bunri University, Kagawa, Japan. maruyama@kph.bunri-u.ac.jp
34. Novel non-nucleoside human cytomegalovirus inhibitors based upon TSAO nucleoside derivatives: structure-activity relationships. Year Published: 2007
35. Synthesis, anticancer, and cytotoxic activities of some mononuclear Ru(II) compounds. Year Published: 2007
Department of Pharmaceutical Chemistry, KLES College of Pharmacy, 2nd Block, Rajajinagar, Bangalore 560010, Karnataka, India. subhasskarki@hotmail.com
36. Targeting platelet-derived endothelial cell growth factor/thymidine phosphorylase for cancer therapy. Year Published: 2007
Laboratory of Virology and Chemotherapy, Rega Institute for Medical Research, K.U. Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium. sandra.liekens@rega.kuleuven.be
37. Mitochondrial expression of the Drosophila melanogaster multisubstrate deoxyribonucleoside kinase. Year Published: 2007
Karolinska Institute, Department of Laboratory Medicine, Division of Clinical Virology F68, S-14186 Stockholm, Sweden. nicola.solaroli@ki.se
38. Characterization and structural analysis of novel mutations in human immunodeficiency virus type 1 reverse transcriptase involved in the regulation of resistance to nonnucleoside inhibitors. Year Published: 2007
Department of Experimental Medicine, University of Rome Tor Vergata, Via Montpellier 1, 00133 Rome, Italy. ceccherini@med.uniroma2.it
39. Ester prodrugs of cyclic 1-(S)-[3-hydroxy-2-(phosphonomethoxy)propyl]-5-azacytosine: synthesis and antiviral activity. Year Published: 2007
Gilead Sciences and IOCB Research Centre, Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic. marcela@uochb.cas.cz
40. Non-nucleoside HIV-1 reverse-transcriptase inhibitors. Part 10. Synthesis and anti-HIV activity of 5-alkyl-6-(1-naphthylmethyl)pyrimidin-4(3H)-ones with a mono- or disubstituted 2-amino function as novel 'dihydro-alkoxy-benzyl-oxopyrimidine' (DABO) analogues. Year Published: 2008
Department of Chemistry, Fudan University, Shanghai 200433, PR China.
41. Synthesis, structural characterization, and biological studies of new antimony(III) complexes with thiones. The influence of the solvent on the geometry of the complexes. Year Published: 2007
Section of Inorganic and Analytical Chemistry, Department of Chemistry, University of Ioannina, 45110 Ioannina, Greece.
42. New developments of the "lock-in" modified cycloSal-d4TMPs. Year Published: 2007
Department of Chemistry, Organic Chemistry, Faculty of Science, University of Hamburg, Martin Luther King-Platz 6, 20146 Hamburg, Germany.
43. Alkyne-azide click chemistry mediated carbanucleosides synthesis. Year Published: 2007
44. Cross-metathesis mediated synthesis of new acyclic nucleoside phosphonates. Year Published: 2007
45. Antiviral activity of 3-(3,5-dimethylbenzyl)uracil derivatives against HIV-1 and HCMV. Year Published: 2007
Faculty of Pharmaceutical Sciences at Kagawa Campus, Tokushima Bunri University, Kagawa, Japan. maruyama@kph.bunri-u.ac.jp
46. Novel non-nucleoside human cytomegalovirus inhibitors based upon TSAO nucleoside derivatives: structure-activity relationships. Year Published: 2007
47. Preclinical development of bicyclic nucleoside analogues as potent and selective inhibitors of varicella zoster virus. Year Published: 2007
Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK. mcguigan@cardiff.ac.uk
48. Hydantoin derivatives of L- and D-amino acids: synthesis and evaluation of their antiviral and antitumoral activity. Year Published: 2007
Department of Medicinal Chemistry, Faculty of Pharmacy and Biochemistry, A. Kovaci?a 1, HR-10000 Zagreb, Croatia. zrajic@pharma.hr
49. A p-[18F]fluoroethoxyphenyl bicyclic nucleoside analogue as a potential positron emission tomography imaging agent for Varicella-Zoster virus thymidine kinase gene expression. Year Published: 2007
Molecular Small Animal Imaging Center, Laboratory for Radiopharmacy-Faculty of Pharmaceutical Sciences, Department of Nuclear Medicine, Rega Institute for Medical Research, Katholieke Universiteit Leuven, Belgium.
50. Synthesis and antiviral activity of the carbocyclic analogue of the highly potent and selective anti-VZV bicyclo furano pyrimidines. Year Published: 2007
Welsh School of Pharmacy, Cardiff University, UK.
51. Novel non-nucleoside human cytomegalovirus inhibitors based upon TSAO nucleoside derivatives: structure-activity relationships. Year Published: 2007
Instituto de Química Médica (CSIC), Madrid, Spain.
52. Increased mitochondrial DNA copy-number in CEM cells resistant to delayed toxicity of 2',3'-dideoxycytidine. Year Published: 2008
Karolinska Institute, Division for Clinical Microbiology, Department of Laboratory Medicine, S-141 86 Stockholm, Sweden.
53. 6-Azathymidine-4'-thionucleosides: synthesis and antiviral evaluation. Year Published: 2008
Medicinal Chemistry, Welsh School of Pharmacy, Cardiff University, Cardiff, CF10 3XF, UK.
54. Non-nucleoside HIV-1 reverse-transcriptase inhibitors. Part 10. Synthesis and anti-HIV activity of 5-alkyl-6-(1-naphthylmethyl)pyrimidin-4(3H)-ones with a mono- or disubstituted 2-amino function as novel 'dihydro-alkoxy-benzyl-oxopyrimidine' (DABO) analogues. Year Published: 2008
Department of Chemistry, Fudan University, Shanghai 200433, PR China.
55. A p-[18F]fluoroethoxyphenyl bicyclic nucleoside analogue as a potential positron emission tomography imaging agent for varicella-zoster virus thymidine kinase gene expression. Year Published: 2007
Molecular Small Animal Imaging Center, Laboratory for Radiopharmacy-Faculty of Pharmaceutical Sciences, Department of Nuclear Medicine, Rega Institute for Medical Research, Katholieke Universiteit Leuven, Belgium.
56. Synthesis and antiviral activity of the carbocyclic analogue of the highly potent and selective anti-VZV bicyclo furano pyrimidines. Year Published: 2007
Welsh School of Pharmacy, Cardiff University, UK.
57. Synthesis, anti-HIV-1 activity, and modeling studies of N-3 Boc TSAO compound. Year Published: 2008
58. Synthesis, anti-HIV-1 activity, and modeling studies of N-3 Boc TSAO compound. Year Published: 2008